It seems reasonable to conclude that Toosendanin is a presynaptic blocking agent.
这些结果表明,川一个选择性地用于突触前的肉传递阻遏剂。
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Cocaine increases the release of certain neurotransmitters, but it's biggest effect is blocking reuptake receptors on presynaptic axon terminals, and both actions keep neurotransmitters like dopamine, norepinephrine, and serotonin in the synapse longer and increases their effects.
可卡因促进一些特定神经递质的释放,但最大的作用是阻止突触前神经元终端受体的“”;两种作用都能使得神经递质,如多巴胺、去甲肾上腺素与5-HT,在突触间隙存留时间延长,从而加强他们的作用。